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Lead Optimization

To obtain potent drugs, suitable chemical modifications are done in the molecules with potential ability of being a drug.

This requires the simultaneous optimization of multiple properties and parameters in the chemical compound and is thus a time consuming and not very economic. The modification of the molecule can be done through molecular modeling, structural biology and quantitative structure-activity relationships.

The drug designing and discovery process include the following major steps:

  1. Drug Target Identification
  2. Target Validation
  3. Lead Compound Identification
  4. Lead Optimization
  5. Preclinical And Clinical development
  6. Administration of Drugs
  7. Absorption Of Drugs
  8. Drug Assays
  9. Preservation Of Pharma Product

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